Cannabinoid Receptor
Cannabinoid Receptor
Cannabinoid receptors are currently classified into three groups: central (CB1), peripheral (CB2) and GPR55, all of which are G-protein-coupled. CB1 receptors are primarily located at central and peripheral nerve terminals. CB2 receptors are predominantly expressed in non-neuronal tissues, particularly immune cells, where they modulate cytokine release and cell migration. Recent reports have suggested that CB2 receptors may also be expressed in the CNS. GPR55 receptors are non-CB1/CB2 receptors that exhibit affinity for endogenous, plant and synthetic cannabinoids. Endogenous ligands for cannabinoid receptors have been discovered, including anandamide and 2-arachidonylglycerol.
Cannabinoid Receptor Isoform Specific Products
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Cannabinoid Receptor Inhibitors
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Cannabinoid Receptor Agonists
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Cannabinoid Receptor Antagonists
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Cannabinoid Receptor Activators
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Cannabinoid Receptor Modulators
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Cannabinoid Receptor Chemical
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Cannabinoid Receptor Inducer
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Cannabinoid Receptor Degrader
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Cannabinoid Receptor Controls
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Cannabinoid Receptor Ligands
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Cannabinoid Receptor Produits associés (442)
Produits associés (442)
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Anticorps (1)
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Cannabinoid Receptor Isoform Comparison
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2-(1-(4-Fluorobenzyl)-1H-indol-3-yl)acetic acid
0 ImagesCat. No.: HY-W030120CAS No.: 176204-51-62-(1-(4-Fluorobenzyl)-1H-indol-3-yl)acetic acid is structurally similar to cannabinoid.
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PSB-SB1202
0 ImagesPSB-SB1202 (Compound 21a) is a phenyl coumarin compound. PSB-SB1202 is a CB1/CB2 agonist with EC50 values of 56 and 14 nM, and Ki values of 32 and 49 nM, respectively.
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exo-Tetrahydrocannabivarin
0 ImagesCat. No.: HY-168368CAS No.: 137008-69-6exo-Tetrahydrocannabivarin (Compound 12) is a Δ9,11-THC analogue. exo-Tetrahydrocannabivarin weakly binds to cannabinoid receptors (CB) (IC50: 1.4 μM). exo-Tetrahydrocannabivarin is active on both motor and analgesic aspects in mice.
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Giminabant
0 ImagesCat. No.: HY-111195CAS No.: 890033-57-5Giminabant is a cannabinoid receptor antagonist for veterinary use. Giminabant can be used for the research of metabolic diseases and addiction-related disorders.
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Δ8-THCPA-A
0 ImagesCat. No.: HY-170696CAS No.: 2897582-89-5Synonyms: Δ8-Tetrahydrocannabiphorolic acidΔ8-THCPA-A (Δ8-Tetrahydrocannabiphorolic acid) is structurally similar to known phytocannabinoids.
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Carmagerol
0 ImagesCat. No.: HY-170703CAS No.: 140396-81-2Carmagerol is a phytocannabinoid metabolite.
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8(R)-Hydroxy-9(R)-hexahydrocannabinol
0 ImagesCat. No.: HY-168789CAS No.: 42793-11-38(R)-Hydroxy-9(R)-hexahydrocannabinol, a phytocannabinoid compound, is a metabolite of 9(R)-Hexahydrocannabinol.
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(±)-8'-Hydroxy cannabichromene
0 ImagesCat. No.: HY-170039CAS No.: 132032-41-88'-Hydroxy cannabichromene is a phytocannabinoid metabolite.
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Rimonabant Hydrochloride (Standard)
0 ImagesSynonyms: SR 141716A Hydrochloride (Standard)Rimonabant (Hydrochloride) (Standard) is the analytical standard of Rimonabant (Hydrochloride). This product is intended for research and analytical applications. Rimonabant Hydrochloride (SR 141716A Hydrochloride) is a highly potent and selective central cannabinoid receptor (CB1) antagonist with an Ki of 1.8 nM. Rimonabant Hydrochloride (SR 141716A Hydrochloride) also inhibits Mycobacterial membrane protein Large 3 (MMPL3).
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5-Fluoro PB-22 N-(2-fluoropentyl) isomer
0 ImagesCat. No.: HY-172043CAS No.: 2365471-10-75-Fluoro PB-22 N-(2-fluoropentyl) isomer is a derivative of cannabinoid.
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Tetrahydrocannabiphorol
0 ImagesCat. No.: HY-W775348CAS No.: 54763-99-4Synonyms: THCPTetrahydrocannabiphorol (THCP) is a phytocannabinoid.
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Rimonabant (Standard)
0 ImagesSynonyms: SR141716 (Standard)Rimonabant (Standard) is the analytical standard of Rimonabant. This product is intended for research and analytical applications. Rimonabant (SR141716) is a highly potent, brain penetrated and selective central cannabinoid receptor (CB1) antagonist with a Ki of 1.8 nM. Rimonabant (SR141716) also inhibits Mycobacterial membrane protein Large 3 (MMPL3).
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CH-PIATA
0 ImagesCat. No.: HY-W728163CAS No.: 3085600-43-4CH-PIATA is a synthetic cannabinoid with an acetamide linker. CH-PIATA can be detected as parent substance in blood samples. CH-PIATA has EC50 values of >71 and >176 nM for CB1 and CB2, respectively.
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Δ9-Tetrahydrocannabiorcol
0 ImagesCat. No.: HY-168817CAS No.: 22972-65-2Δ9-Tetrahydrocannabiorcol is structurally similar to known phytocannabinoids.
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Δ9-THCH
0 ImagesCat. No.: HY-168813CAS No.: 36482-24-3Δ9-THCH is structurally similar to known phytocannabinoids.
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AM281 (Standard)
0 ImagesCat. No.: HY-13505RCAS No.: 202463-68-1
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(±)-CBCP
0 ImagesCat. No.: HY-170726CAS No.: 55824-16-3Synonyms: (±)-Cannabichromephorol(±)-CBCP ((±)-Cannabichromephorol) is structurally similar to known phytocannabinoids.
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RTI-371
0 ImagesCat. No.: HY-129215CAS No.: 652978-45-5RTI-371 is a highly selective atypical dopamine transporter (DAT) inhibitor that crosses the blood-brain barrier. RTI-371 exhibits potent inhibitory activity in cell lines transfected with human DAT (IC50 = 8.7 nM) and shows high binding affinity for rat DAT with a Ki value of 7.81 nM. RTI-371 also acts as a positive allosteric modulator of the human cannabinoid 1 receptor (hCB1 receptor), enhancing the activity of cannabinoid receptor agonists in a concentration-dependent manner. RTI-371 can be used for the research of Parkinson's disease.
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Cannabicyclolic acid
0 ImagesCat. No.: HY-W775308CAS No.: 40524-99-0Cannabicyclolic acid is a certified reference material categorized as a photodegradation product of the phytocannabinoid Cannabichromenic acid.
